Nature.com April 29, 2026 • 22:07

GLP-1R–GIPR–PPARα/γ/δ quintuple agonism corrects obesity and diabetes in mice - Nature

GLP-1R–GIPR–PPARα/γ/δ quintuple agonism corrects obesity and diabetes in mice - Nature

GLP-1–GIP–lanifibranor, a single-molecule agonist of GLP-1R, GIPR, PPARα, PPARγ and PPARδ, shows promising therapeutic efficacy against obesity-linked metabolic dysfunction in vitro and in mouse models via synergistic incretin and PPAR activity.

Animals and housing conditions
Experiments were performed in accordance with the Animal Protection Law of the European Union after permission by the Governments of Upper Bavaria, Germany, or Copenha… [+11715 chars]

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